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publicationDate 2014-07-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2014108452-A1
titleOfInvention Proteolysis targeting chimeras (protacs) directed to the modulation of the estrogen receptor
abstract A compound of formula (I): or a pharmaceutically acceptable salt thereof, compositions, combinations and medicaments containing said compounds and processes for their preparation. The invention also relates to the use of said compounds, combinations, compositions and medicaments, for example as inhibitors of the activity of the estrogen receptor, including degrading the estrogen receptor, the treatment of diseases and conditions mediated by the estrogen receptor.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C9E1
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Total number of triples: 1332.