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publicationDate 2020-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10865202-B2
titleOfInvention Indole derivatives as estrogen receptor degraders
abstract The present disclosure relates to compounds and a pharmaceutically acceptable salt thereof, compositions, combinations and medicaments containing the compounds, and processes for their preparation. The disclosure also relates to the use of the compounds, combinations, compositions and medicaments, for example as inhibitors of the activity of the estrogen receptor, including degrading the estrogen receptor, the treatment of diseases and conditions mediated by the estrogen receptor.
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Total number of triples: 3127.