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publicationDate 2017-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9632089-B2
titleOfInvention Small-molecule hydrophobic tagging of fusion proteins and induced degradation of same
abstract The present invention includes compounds that are useful in perturbing or disrupting the function of a transmembrane or intracellular protein, whereby binding of the compounds to the transmembrane or intracellular protein induces proteasomal degradation of the transmembrane or intracellular protein. The present invention further includes a method of inducing proteasomal degradation of a transmembrane or intracellular protein. The present invention further includes a method of identifying or validating a protein of interest as a therapeutic target for treatment of a disease state or condition.
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Total number of triples: 1480.