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publicationDate 2011-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2011100401-A1
titleOfInvention Macrocycles as factor xia inhibitors
abstract The present invention provides compounds of Formula (I): or a stereoisomer, a tautomer, or a pharmaceutically acceptable salt thereof, wherein all the variables are as defined herein. These compounds are selective Factor XIa inhibitors or dual inhibitors of fXIa and plasma kallikrein. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating thromboembolic and/or inflammatory disorders using the same.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP45643
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25273605
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419656966
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID75771
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237435619
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP45654
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08591

Total number of triples: 5621.