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filingDate 2016-07-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5fa35544ee14f95e8378803188d1eaba
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publicationDate 2019-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10287288-B2
titleOfInvention Factor XIa macrocyclic inhibitors bearing alkyl or cycloalkyl P2' moieties
abstract The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compounds are selective factor XIa inhibitors or dual inhibitors of FXIa and plasma kallikrein. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating thromboembolic and/or inflammatory disorders using the same.
priorityDate 2015-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1865.