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filingDate 2015-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f4ee67145e738aea5694aa6c8529f312
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publicationDate 2018-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10081623-B2
titleOfInvention Diamide macrocycles that are FXIa inhibitors
abstract The present invention provides compounds of Formula (I) or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compounds are selective Factor XIa inhibitors or dual inhibitors of FXIa and plasma kallikrein. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating thromboembolic and/or inflammatory disorders using the same.
priorityDate 2014-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284371
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID564868
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Total number of triples: 1303.