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publicationNumber US-11142508-B2
titleOfInvention Bisphenol derivatives and their use as androgen receptor activity modulators
abstract Compounds having a structure of Formula Ior a pharmaceutically acceptable salt, tautomer or stereoisomer thereof, wherein R1, R2, R3, R11a, R11b, R11c, R11d, and X, are as defined herein, are provided. Uses of such compounds for modulating androgen receptor activity, imaging diagnostics in cancer and therapeutics, and methods for treatment of subjects in need thereof, including prostate cancer are also provided.
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Total number of triples: 3096.