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publicationDate 2017-10-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2017298033-A1
titleOfInvention Bisphenol derivatives and their use as androgen receptor activity modulators
abstract Compounds having a structure of Formula I: n n n n n n n n n n or a pharmaceutically acceptable salt, tautomer or stereoisomer thereof, wherein R 1 , R 2 , R 3 , R 11a , R 11b , R 11c , R 11d , and X, are as defined herein, are provided. Uses of such compounds for modulating androgen receptor activity, imaging diagnostics in cancer and therapeutics, and methods for treatment of subjects in need thereof, including prostate cancer are also provided.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026755
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157832541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978967
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026756
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7582
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978968
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450093069
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026749
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978977
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026750
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978978
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450096798
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026751
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132007351
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026752
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978979
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132007352
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026762
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978980
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID353978973
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132026763

Total number of triples: 3435.