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filingDate 2019-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-10-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1d74d01a19ac18c2188d09177a504cc0
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publicationDate 2020-10-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10807982-B2
titleOfInvention Bromodomain inhibitors
abstract The present invention relates to substituted heterocyclic derivative compounds, compositions comprising said compounds, and the use of said compounds and compositions for epigenetic regulation by inhibition of bromodomain-mediated recognition of acetyl lysine regions of proteins, such as histones. Said compositions and methods are useful for the treatment of cancer and neoplastic disease.
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Total number of triples: 2368.