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publicationDate 2016-05-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2016077378-A1
titleOfInvention Substituted pyrrolopyrdines as inhibitors of bromodomain
abstract The present invention relates to compounds of formula (I) and to salts thereof, wherein R 1 , R 2 , and Q have any of the values defined in the specification, and compositions and uses thereof. The compounds are useful as inhibitors of bromodomains. Also included are pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various bromodomain-mediated disorders.
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Total number of triples: 3907.