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filingDate 2016-04-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ee0404c15025a946729fede453f951b2
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publicationDate 2017-02-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2017050968-A1
titleOfInvention Bromodomain inhibitor
abstract The present invention relates to substituted heterocyclic derivative compounds, compositions comprising said compounds, and the use of said compounds and compositions for epigenetic regulation by inhibition of bromodomain-mediated recognition of acetyl lysine regions of proteins, such as histones. Said compositions and methods are useful for the treatment of cancer and neoplastic disease.
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Total number of triples: 2410.