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filingDate 2017-02-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-07-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f7e2f0ae6eceef6d8a7ec19e45c37eef
publicationDate 2018-07-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10023592-B2
titleOfInvention Bromodomain inhibitors
abstract The present invention relates to substituted heterocyclic derivative compounds, compositions comprising said compounds, and the use of said compounds and compositions for epigenetic regulation by inhibition of bromodomain-mediated recognition of acetyl lysine regions of proteins, such as histones. Said compositions and methods are useful for the treatment of cancer and neoplastic disease.
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priorityDate 2013-10-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 6143.