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publicationDate 2008-10-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2008119741-A2
titleOfInvention 3-imidazolyl-indoles for the treatment of proliferative diseases
abstract The invention relates to 3-heterocyclyl indolyl compounds capable of inhibiting the interaction between p53, or variants thereof, and MDM2 and/or MDM4, or variants thereof, respectively, said compounds having the formula (I) wherein R1, R2, R3, R4, RA, Y and Y are as defined in the specification. Due to their activity, the compounds are useful in the treatment of various disorders and diseases mediated by the activity of MDM2 and/or MDM4, or variants thereof, such as inflammatory or proliferative diseases or in the protection of cells.
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Total number of triples: 4240.