http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2018015558-A1

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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2f53ecd13289222aa80a274d0511e690
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publicationDate 2018-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2018015558-A1
titleOfInvention Imidazolyl-substituted indole derivatives binding 5-ht7 serotonin receptor and pharmaceutical compositions thereof
abstract The invention relates to a new class of substituted indole derivatives that are able to activate 5-HT 7 serotonin receptor. These compounds bind 5-HT 7 serotonin receptor with high affinity and selectivity, while possessing favourable physicochemical properties. The compounds of the invention are the first described low-basicity 5-HT 7 receptor agonists. The invention also relates to use of such compounds in the treatment or prevention of 5-HT 7 receptor-related disorders, especially of the central nervous system. The invention also relates to the isotopically labelled compounds for use in the in vivo diagnostics or imaging of a 5-HT 7 serotonin receptor.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134188365
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423403
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227337546
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134188362
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450216206
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10256
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146229
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138691355
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416193197
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393293
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID141631929
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID141631930
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417702
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138691364
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87894
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392451
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID141631933
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415940483
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1833
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405609
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138691362
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394734
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID141631931
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID141631932
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415772768
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226580841
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227338745
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226943536
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138691366
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID27513
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153993173
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394295
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138691340
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226426880
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11978
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449603119
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2774502
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1001
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18476134

Total number of triples: 354.