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filingDate 2002-10-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-04-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03032981-A1
titleOfInvention 4-(4-alkoxy-3-hydroxyphenyl)-2-pyrrolidone derivatives as pde-4 inhibitors for the treatment of neurological syndromes
abstract Selective PDE4 inhibition is achieved by 4-(substituted-phenyl)-2-pyrrolidinone compounds. The compounds exhibit improved PDE4 inhibition as compared to compounds like rolipram and show selectivity with regard to inhibition of other classes of PDEs. The compounds of the present invention are of formula (I), wherein R1, R2 and R3 are as defined herein.
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Total number of triples: 1523.