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grantDate 2017-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b17fa8ce177fb58c2a8258489e9304b2
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publicationDate 2017-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9670181-B2
titleOfInvention Substituted 6,7-dialkoxy-3-isoquinolinol derivatives as inhibitors of phosphodiesterase 10 (PDE 10A)
abstract The invention relates to compounds of the formula n nwherein R′, R 1 through R 7 and Ar are as defined herein. These compounds are useful as inhibitors of phosphodiesterase 10 (PDE10A) which are useful in treating central nervous system diseases such as psychosis and also in treating, for example, obesity, type II diabetes, metabolic syndrome, glucose intolerance, pain and ophthalmic diseases.
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Total number of triples: 2141.