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publicationNumber US-9439912-B2
titleOfInvention Androgen receptor down-regulating agents and uses thereof
abstract The present disclosure provides the design and synthesis of novel steroidal compounds that cause down-regulation of the androgen receptor (AR), both full length and splice variant. The compounds are potential agents for the treatment of all forms of prostate cancer and other diseases that depend on functional AR.
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Total number of triples: 812.