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publicationDate 2003-07-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6586434-B2
titleOfInvention Method for the preparation of tetrahydrobenzothiepines
abstract Among its several embodiments, the present invention provides an improved process for the preparation of tetrahydrobenzothiepine-1,1-dioxide compounds; the provision of a process for preparing a diastereomeric mixture of tetrahydrobenzothiepine-1,1-dioxide compounds from a single diastereomer of such compounds; the provision of a process for the preparation of 3-bromo-2-substituted propionaldehyde compounds; and the provision of a process for the preparation of 3-thio-2-substituted propionaldehyde compounds.
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Total number of triples: 1409.