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titleOfInvention Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
abstract Provided are novel benzothiepines, derivatives, and analogs thereof; pharmaceutical compositions containing them; and methods of using these compounds and compositions in medicine, particularly in the prophylaxis and treatment of hyperlipidemic conditions such as those associated with atherosclerosis or hypercholesterolemia, in mammals.
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Total number of triples: 4314.