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publicationNumber US-6258782-B1
titleOfInvention Hybrid polypeptides with enhanced pharmacokinetic properties
abstract The present invention relates to enhancer peptide sequences originally derived from various retroviral envelope (gp41) protein sequences that enhance the pharmacokinetic properties of any core polypeptide to which they are linked. The invention is based on the discovery that hybrid polypeptides comprising the enhancer peptide sequences linked to a core polypeptide possess enhanced pharmacokinetic properties such as increased half life. The invention further relates to methods for enhancing the pharmacokinetic properties of any core polypeptide through linkage of the enhancer peptide sequences to the core polypeptide. The core polypeptides to be used in the practice of the invention can include any pharmacologically useful peptide that can be used, for example, as a therapeutic or prophylactic reagent.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457757
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211421
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455358
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485217942
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211306
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457759
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485212792
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485215596
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455367
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145456814
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9841219
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444446
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485214848
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455375
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9841671
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211314
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485221170
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455128
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211292
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403335
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455136
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457096
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457791
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID77844313
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485221176
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485215515
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485213116
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211295
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457793
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145454994
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444128
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID232
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211298
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485221082
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44608124
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457795
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485222770
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485221083
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485214886
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44610015
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485217928
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485212444
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457797
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426419098
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485215498
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419540617
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485211301
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485217931
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485212446
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457799
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485212447
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457778
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485221092
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455042
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145456828
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25002196
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455003
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145457781
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145455072
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID485212450

Total number of triples: 4104.