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publicationNumber US-5693648-A
titleOfInvention O-aryl, O-alkyl, O-alkenyl and O-alkynyl-macrolides having immunosuppressive activity
abstract PCT No. PCT/US94/11114 Sec. 371 Date Mar. 27, 1996 Sec. 102(e) Date Mar. 27, 1996 PCT Filed Sep. 30, 1994 PCT Pub. No. WO95/09857 PCT Pub. Date Apr. 13, 1995Substituted compounds of the FK-506 Type. These compounds are useful for the same or essentially the same purposes as FK-506 and are applied in the same or a similar manner. These compounds are immunosuppressants and useful for the treatment of autoimmune diseases, infectious diseases and/or the prevention of rejection of foreign organ transplants. Still other uses are described in the disclosure.
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Total number of triples: 1106.