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publicationNumber US-2006058323-A1
titleOfInvention New 8-(3-amino-piperidin-1-yl)-7-(but-2-ynyl)-xanthines, the preparation thereof and their use as pharmaceutical compositions
abstract The application relates to new substituted xanthines of general formula n n nwherein R 1 and R 2 are defined as in claims 1 to 11 , the tautomers, the enantiomers, the diastereomers, the mixtures thereof and the salts thereof, which have valuable pharmacological properties, particularly an inhibiting effect on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).
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Total number of triples: 1376.