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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c92b7f6e9f50c24b55ecf716e6dc51ee
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publicationDate 2005-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2005130985-A1
titleOfInvention 8-(piperazin-1yl)- and 8-([1,4]diazepan-1yl)-xanthines, the preparation thereof and their use as pharmaceutical composition
abstract The present invention relates to substituted xanthines of the general formula n n nin which R 1 to R 3 and n are as defined in claims 1 to 8, their tautomers, their enantiomers, their diastereomers, their mixtures, their prodrugs and their salts, which have valuable pharmacological properties, in particular an inhibitory action on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).
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Total number of triples: 587.