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publicationDate 2005-02-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2005026921-A1
titleOfInvention New imidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
abstract The present invention relates to substituted imidazo-pyridinones and imidazo-pyridazinones of general formula n n nwherein Y and R 1 to R 4 are defined as in claim 1, the tautomers, enantiomers, diastereomers, the mixtures thereof and the salts thereof, which have valuable pharmacological properties, particularly an inhibiting effect on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).
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Total number of triples: 1498.