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filingDate 2020-03-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-02-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a8a76b5e9e69ff461530d2bdb5a02b7e
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publicationDate 2022-02-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11254672-B2
titleOfInvention Dihydrobenzimidazolones for medical treatment
abstract The present invention provides selected dihydrobenzimidazolones which bind to the ubiquitously expressed E3 ligase protein cereblon (CRBN) and alter the substrate specificity of the CRBN E3 ubiquitin ligase complex, resulting in breakdown of intrinsic downstream proteins. The disclosed compounds are useful for the treatment of cancer.
priorityDate 2017-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1643.