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filingDate 2016-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-10-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d68d9cca34a38edcb4d1d0d093936827
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publicationDate 2021-10-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11147771-B2
titleOfInvention Orodispersible dosage unit containing an estetrol component
abstract The invention provides an orodispersible solid pharmaceutical dosage unit having a weight between 30 and 1,000 mg, said dosage unit consisting of: 0.1-25 wt. % of estetrol particles containing at least 80 wt. % of an estetrol component selected from estetrol, estetrol esters and combinations thereof; and 75-99.9 wt. % of one or more pharmaceutically acceptable ingredients; the solid dosage unit comprising at least 100 μg of the estetrol component; and wherein the solid dosage unit can be obtained by a process comprising wet granulation of estetrol particles having a volume weighted average particle size of 2 μm to 50 μm. The solid dosage unit is easy to manufacture and perfectly suited for sublingual, buccal or sublabial administration.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6917715
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65157
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6238
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226426036
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396046
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226412118
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6128
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396047
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399858
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414984
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6230
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107428
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20415
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423122
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423106
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6231
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396137
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ62588
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20848881
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393698
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396146
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284557
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408624
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393714
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25249
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396147
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408625
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396114
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID27125
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009224
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68873
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226507690
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID40973
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID138043
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396927
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9949848
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396115
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226426035
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP97497
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135413523
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226633472
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226422998
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226506936
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5991
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226626651
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID228864
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405588
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6251
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226426388
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5995
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24775
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5994
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423123
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6540478
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226666481
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9270
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226666480
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5984
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0EQL2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226666482
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399998
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9842127
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID138043
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID103023
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393830
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6607
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227201854
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66577627
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423270
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID51066490
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6462
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14743
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226512788
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10953859
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7427
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226412813
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405557
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10476437

Total number of triples: 373.