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filingDate 2016-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2019-03-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10238647-B2
titleOfInvention Compositions for affecting weight loss
abstract Disclosed are compositions for affecting weight loss comprising a first compound and a second compound, where the first compound is an opioid antagonist and the second compound causes increased agonism of a melanocortin 3 receptor (MC3-R) or a melanocortin 4 receptor (MC4-R) compared to normal physiological conditions. Also disclosed are methods of affecting weight loss, increasing energy expenditure, increasing satiety in an individual, or suppressing the appetite of an individual, comprising identifying an individual in need thereof and treating that individual to antagonize opioid receptor activity and to enhance α-MSH activity.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410554594
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393293
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PJB2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743275
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405584
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100533423
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ98TA8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865X8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100136771
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226420049
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395015
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743278
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ63264
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5311017
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395016
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30487
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100052414
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507197
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507269
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01203
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493269
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419580638
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6093260
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397763
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393271
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68200185
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493286
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447968746
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554909
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455400546
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226432808
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419497074
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XSW9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397563
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503199
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XS77
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01308
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5734
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393518
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9NDE7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554878
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426147153
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2130
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9N2C1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226449465
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3081925
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID548631
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5443
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91082
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396158
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60961
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3549980
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7098641
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID38065
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419555613
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414500
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25569
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414425
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6476
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID22044
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399686
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7582
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID181
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5078
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414681
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403974
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45051774
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48090
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107428
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414652
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP79182
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID561647
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5361918
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJU0

Total number of triples: 982.