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publicationNumber RU-2460724-C2
titleOfInvention Substituted arylimidazolones and triazolones as vasopressin receptor inhibitors
abstract FIELD: chemistry. n SUBSTANCE: described are novel 1,2,4-triazolones of general formula (I): n , where A denotes N and values of other radicals are given in the claim, which are vasopressin receptor inhibitors, synthesis method thereof and use thereof to prepare medicinal agents for treating and/or preventing diseases, particularly for treating and/or preventing cardiovascular diseases. n EFFECT: high efficiency of using said derivatives. n 6 cl, 512 ex
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