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filingDate 2005-09-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2011-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2397563-A2
titleOfInvention Enhanced antisense oligonucleotides
abstract Described herein are gap-widened antisense oligonucleotides having improved therapeutic index as compared to 5-10-5 MOE gapmer antisense oligonucleotides of the same sequence. Also described are methods of reducing a target RNA in an animal using the gap-widened antisense oligonucleotides of the present invention. Further, are methods for selecting a gap-widened antisense oligonucleotides.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO70372
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9YFS9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ94818
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0R2M2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5ULT9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8625716
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396842
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226520094
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83601
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID252900
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A0H3MAB5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID553740
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22947699
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID33824
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19315
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19314
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP12245
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID35799
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9PJN6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID317743
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6URW1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID35728
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DB19
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226434183
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24383
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DB18
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04797
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ07203
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129901274
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6UUN9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128632074
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2NEN0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ673L6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID368415
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13050061
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23722
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19593
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226588339
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421319801
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416216707
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6L125
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID243308914
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49262
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449204649
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5728
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128686785
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49254
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID455722
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID66824
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507980
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ01651
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID459934
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04406
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5V061
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1PS67
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WN83
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WN82
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A038
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1YD06
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP32809
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A1P1
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226610180
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID74857
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID92918
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4KHW5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ64467
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Total number of triples: 465.