http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022187417-A1

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filingDate 2022-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7a1c9ee0c8fce3110919ba418e047cd6
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publicationDate 2022-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022187417-A1
titleOfInvention Small molecule degraders of cbp/p300 proteins
abstract The present disclosure relates to compounds of Formula (I):, and the pharmaceutically acceptable salts and solvates thereof, wherein A, m, X, Y, Z, and B 1 are as defined as set forth in the specification. The present disclosure also relates to uses of the compounds, e.g., in treating or preventing a condition or disorder responsive to the degradation of CBP/P300 proteins (e.g., cancer).
priorityDate 2021-03-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43428
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416226230
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452185578
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419500669
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3874950
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492980
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID564470
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394985
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119236
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID238
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A3Q1MKE9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419487788
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8119
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148195
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501828
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16542
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393601
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID481558
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428401474
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID566841
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421334983
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450594909

Total number of triples: 652.