http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019121670-A1

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filingDate 2018-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e908361c478b972e28978ed5be137029
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publicationDate 2019-06-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019121670-A1
titleOfInvention 4,5-dihydro-1h-thieno[2,3-g]indazolyl derivatives having multimodal activity against pain
abstract wherein the meanings for the various substituents are as disclosed in the description, having dual pharmacological activity towards both the α2δ subunit, in particular the α2δ-1 subunit, of the voltage-gated calcium channel and the μ-opioid receptor, to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy, in particular for the treatment of pain.
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Total number of triples: 371.