http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019060536-A1

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filingDate 2018-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e3d8ad206f8ddce84cca5393d5eaa348
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d6630818aed76605112c1f8ca0ecc2a5
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publicationDate 2019-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2019060536-A1
titleOfInvention CO-CRYSTALLINE FORMS OF ((1S, 2S, 4R) -4- {4 - [(1S) -2,3-DIHYDRO-1H-INDEN-1-YLAMINO] -7H-PYRROLO [2,3-D] PYRIMIDIN -7-YL} -2-HYDROXYCYCLOPENTYL) METHYLSULFAMATE, THEIR FORMULATIONS AND USES
abstract The present invention relates to co-crystalline forms of ((1S, 2S, 4R) -4- {4 - [(1S) -2,3-dihydro-1H-inden-1-ylamino] -7H-pyrrolo [2, 3-d] pyrimidin-7-yl} -2-hydroxycyclopentyl) methylsulfamate of formula ( I ). The invention also relates to methods for producing (15S, 2S, 4R) -4- {4 - [(1S) -2,3-dihydro-1H-inden-1-ylamino] -7H-pyrroloacocrystalline forms of [2,3-d] pyrimidin-7-yl} -2-hydroxycyclopentyl) methylsulfamate of formula ( I ). The invention also relates to the pharmaceutical use of a co-crystalline form as an activating enzyme inhibitor E1, as well as a pharmaceutical composition comprising said co-crystalline form. A method of treatment comprising administering a co-crystalline form of ((1S, 2S, 4R) -4- {4 - [(1S) -2,3-dihydro-1H-inden-1-ylamino] 7H-pyrrolo [2,3-d] pyrimidin-7-yl} -2-hydroxycyclopentyl) methylsulfamate of formula ( I ) is further described.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-11124519-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022112951-A1
priorityDate 2017-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 452.