http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-11124519-B2

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_fd47318319f20f7f99d9fef1fd3e511b
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-13
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-519
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04
filingDate 2018-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ebc9c6a2feff48f19f37153ae8c833a2
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e3d8ad206f8ddce84cca5393d5eaa348
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d6630818aed76605112c1f8ca0ecc2a5
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f2fb2a795b4c7ec9c0d9309a8fd1e9ba
publicationDate 2021-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11124519-B2
titleOfInvention Cocrystal forms of ((1S,2S,4R)-4-{4-[(1S)-2,3-dihydro-1H-inden-1-ylamino]-7H-pyrrolo [2,3-d]pyrimidin-7-yl}-2-hydroxycyclopentyl) methyl sulfamate, formulations and uses thereof
abstract The present invention is directed to cocrystal forms of ((1S,2S,4R)-4-{4-[(1S)-2,3-dihydro-1H-inden-1-ylamino]-7H-pyrrolo[2,3-d]pyrimidin-7-yl}-2-hydroxcyclopentyl) methyl sulfamate of formula (I). The invention is also directed to methods of making cocrystal forms of ((1S,2S,4R)-4-{4-[(1S)-2,3-dihydro-1H-inden-1-ylamino]-7H-pyrrolo[2,3-d]pyrimidin-7-yl}-2-hydroxycyclopentyl) methyl sulfamate of formula (I). The invention is also directed to the pharmaceutical use of a cocrystal form as an E1 activating enzyme inhibitor, as well as a pharmaceutical composition comprising a cocrystal form. The invention is further directed to a method of treatment comprising administering a cocrystal form of ((1S,2S,4R)-4-{4-[(1S)-2,3-dihydro-1H-inden-1-ylamino]-7H-pyrrolo [2,3-d]pyrimidin-7-yl}-2-hydroxycyclopentyl)methyl sulfamate of formula (I).
priorityDate 2017-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2012258977-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2017136024-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2019060536-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2006189636-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2007092213-A2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9827246-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2012258927-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2015164901-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2015030601-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2009036678-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9187482-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2011021544-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2013289037-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-8207177-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2017107579-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10662477-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014055543-A2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2017105995-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9962386-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10745404-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2016030432-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-8933225-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9683003-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2007191293-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2019255052-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9802938-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2016004136-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2013052814-A2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2020085821-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10016427-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2015119410-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2009042013-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2013063481-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2013063496-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2010132110-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10335410-B2
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57417070
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6335613
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5281078
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396360
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399573
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31703
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66577526
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2478
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID460612
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5668
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID439079072
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399572
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65041
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395931
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394128
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID439079077
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226398204
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1292
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID439079062
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396332
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3690
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID439079064
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID445643
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2019
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3469
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396322
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394094
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID439079061
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395671
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394721
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394073
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395672
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5426
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395921
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4054
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396105
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395167
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148124
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396306
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394688
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284623
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID445639
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395166
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30751
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284558
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395655
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395632
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID643460
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2708
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394017
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399463
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7914
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395153
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396074
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5865
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397441
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395394
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136123990
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395888
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395395
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID452548
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16218600
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395152
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9651
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396057
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4212
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395881
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4112
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7059415
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3950
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395574
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395874
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396779
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID29327
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284616
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8567
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395875
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395122
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396493
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID443939
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID657237
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395865
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID77991
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396787
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393970
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395857
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66628257
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396492
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393971
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45051774
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426344796
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395352
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397214
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396287
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395070
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2682
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5364430
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396288
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID384705923
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396480
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284373
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396483
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57417230
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5198
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395069
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5363269
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397955
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID464
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393904
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5746
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID457193
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444539
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60750
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5394
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126941
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID42890
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2907
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8042
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5143
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1263681
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393830
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID64780
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5339
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393293
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394314
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394993
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397122
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396689
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393829
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397123
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID357772
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21414
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396241
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395836
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394280
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID637517
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135403648
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4049
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21584252
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226398946
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396435
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395834
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397695
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396436
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226552040
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395835
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123631
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60700
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226398866
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396679
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226402942
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2265
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5743
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395833
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396002
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30323
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395817
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID36462
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123596
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14455022
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396419
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396001
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397589
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226412273
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21491
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2578
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395512
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396417
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID244
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226582933
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155075219
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1183
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135197385
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23676745
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID219463
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5291
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155075217
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395791
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60838
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395292
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155075215
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395777
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6253
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397529
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155075216
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24360
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID231224
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID249332
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5978
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57068419
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155075214
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16720766
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395968
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11177
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394900
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5453
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396384
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226421438
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID36314
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8892
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395470
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395948
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID439693
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395471
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID243
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395940

Total number of triples: 265.