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filingDate 2017-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_da3044eac224813411b3ef868c3e1c9f
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publicationDate 2018-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2018103663-A1
titleOfInvention Substituted pyrazinecarboxamide compound and composition comprising same and use thereof
abstract Provided in the present invention are a substituted pyrazinecarboxamide compound and a composition comprising the same and the use thereof. The substituted pyrazinecarboxamide compound is a pyrazinecarboxamide compound as represented by formula (I), or a crystal form, a pharmaceutically acceptable salt, a prodrug, a stereoisomer, a hydrate or a solvate thereof. The substituted pyrazinecarboxamide compound and the composition comprising the same disclosed in the present invention have excellent inhibition on an EGFR kinase, and moreover have better pharmacokinetic parametric properties, and can raise the drug concentration of the compound in the animal bodies so as to improve drug efficacy and safety.
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priorityDate 2016-12-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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