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filingDate 2013-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2013-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2013158262-A1
titleOfInvention Ring constrained analogs as arginase inhibitors
abstract The inventive boronic acid analogs are potent inhibitors of Arginase I and II activity. These compounds are candidate therapeutics for treating a disease or disorder associated with an imbalance in the activity or concentration of cellular arginase I and arginase II enzymes. The invention also provides pharmaceutical compositions of the inventive compounds and methods for using the compositions for therapy.
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Total number of triples: 807.