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publicationDate 2012-05-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2012058065-A1
titleOfInvention Boronates as arginase inhibitors
abstract Compounds according to Formula I are potent inhibitors of Arginase I and II activity: (I) where R 1 , R 2 , R 3 , R 4 , D, W, X, Y, and Z are defined in the specification. The invention also provides pharmaceutical compositions of the compounds and methods of their use in treating or preventing a disease or a condition associated with arginase activity.
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Total number of triples: 2095.