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publicationDate 2011-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2011137320-A2
titleOfInvention Small molecule inhibitors of usp1 deubiquitinating enzyme activity
abstract Provided are small molecule inhibitors of ubiquitin specific protease 1 (USP1) activity and methods for their use in treating and characterizing cancers. The small molecule USP1 inhibitors of the invention are particularly useful in the treatment of cancers that are resistant to DNA cross-linking agents.
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Total number of triples: 1710.