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grantDate 2017-08-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3927d006f413ac30a8a8678a305d6482
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publicationDate 2017-08-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9725425-B1
titleOfInvention Compounds and methods for treating cancer
abstract Provided are small molecule inhibitors of ubiquitin specific protease 2, 8 and 12 (USP2 and USP8 and USP12) activity and methods for their use in treating cancers. The small molecule inhibitors of the invention are particularly useful in the treatment of non-small cell lung cancers that are resistant to tyrosine kinase inhibitors and in the treatment of prostate cancer that is resistant to AR inhibitor therapy.
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Total number of triples: 1426.