http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2009058734-A4

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filingDate 2008-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d50369748615e489e53a235de3e68f9e
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publicationDate 2009-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2009058734-A4
titleOfInvention Compounds exhibiting glucagon antagonist and glp-1 agonist activity
abstract Glucagon analogs are disclosed that exhibit both glucagon antagonist and GLP-1 agonist activity. In one embodiment, the glucagon antagonist/GLP-1 agonist comprises a modified amino acid sequence of native glucagon, in which the first one to five N-terminal amino acids of native glucagon is deleted and in which the alpha helix is stabilized.
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