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filingDate 2009-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2015-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8969288-B2
titleOfInvention Amide based glucagon and superfamily peptide prodrugs
abstract Prodrug formulations of glucagon superfamily peptides are provided wherein the glucagon superfamily peptide has been modified by the linkage of a dipeptide to the glucagon superfamily through an amide bond linkage. The prodrugs disclosed herein have extended half lives and are converted to the active form at physiological conditions through a non-enzymatic reaction driven by chemical instability.
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Total number of triples: 2620.