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publicationDate 2008-10-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2008118724-A1
titleOfInvention Indole carboxamides as ikk2 inhibitors
abstract The invention is directed to novel indole carboxamide compounds. Specifically, the invention is directed to compounds according to formula (I): wherein R1, R2, R3, R4, and m are as defined herein. The compounds of the invention are inhibitors of IKK2 and can be useful in the treatment of disorders associated with inappropriate IKK2 (also known as IKKβ) activity, such as rheumatoid arthritis, asthma, rhinitis, and COPD (chronic obstructive pulmonary disease). Accordingly, the invention is further directed to pharmaceutical compositions comprising a compound of the invention. The invention is still further directed to methods of inhibiting IKK2 activity and treatment of disorders associated therewith using a compound of the invention or a pharmaceutical composition comprising a compound of the invention.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332744
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332743
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332726
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451679761
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19861
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12609719
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID43232
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332725
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12335978
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332724
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421888096
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332723
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534753
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412231773
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403113
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397086
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332720
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332719
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332734
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419883798
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP56492
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332733
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127697018
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332732
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID285645
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8CX28
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414893734
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332730
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12443366
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129886338
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394438
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332729
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114461
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409391
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504142
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332727
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129344997
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419577911
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62603004
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128374106
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4SG14
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332773
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394178
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49113
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332772
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226492475
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332771
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332770
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID33036
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332769
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129694219
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129347866
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332783
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127617532
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332782
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419578152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394244
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332781
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332780
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23049600
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332779
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18379236
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332778
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http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID1314
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF4JBP3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF4IRW0
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394773
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60830
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59332755
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7708

Total number of triples: 3820.