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filingDate 2006-07-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ce6d06594f9eaf7a3d9f0a0b9e256d19
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publicationDate 2007-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2007010847-A1
titleOfInvention Sustained release preparation
abstract [PROBLEMS] To provide a preparation which shows a satisfactory gastric residence time, has such a size that is easy to be ingested, can be disintegrated rapidly after the excretion from the stomach, and can be prepared readily in an industrial scale. [MEANS FOR SOLVING PROBLEMS] A gastric retentive preparation having a gastric resident layer and a drug release layer, wherein the gastric resident layer is never disintegrated in the stomach and is disintegrated in the intestine. Preferably, the gastric resident layer shows the minimum diameter of 7 mm or more as measured after stirring the preparation in a first solution at 200 rpm at 37°C for 15 hours under the conditions for the paddle method in the dissolution test in accordance with Japanese Pharmacopoeia and shows the maximum diameter of 6 mm or less as measured after further stirring the preparation in a second solution at 200 rpm at 37°C for 9 hours under the same conditions.
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