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filingDate 2005-08-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8d59c2db1a5344891d20d224d9911280
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publicationDate 2006-03-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2006026430-A2
titleOfInvention Cyclopamine analogues and methods of use thereof
abstract The present invention provides compositions and methods for modulating smoothened­dependent pathway activation. The present invention provides analogs of cyclopamine that can be used to counteract the phenotypic effects of unwanted activation of a hedgehog pathway, such as resulting from hedgehog gain-of-function, Ptc loss-of-function or smoothened gain-of­function mutations. The compounds of the present invention are particularly useful in treating cancers.
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Total number of triples: 870.