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filingDate 2004-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_302226a84e6ed49e1b6f6197383b3679
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publicationDate 2005-04-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2005032468-A2
titleOfInvention Monocyclic and bicyclic lactams as factor xa inhibitors
abstract The present application describes monocyclic and bicyclic lactams and derivatives thereof of Formulae (Ia-e); wherein one of one of T1 and T2 is carbonyl, thiocarbonyl, or sulfonyl or pharmaceutically acceptable salt forms thereof. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.
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Total number of triples: 3316.