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filingDate 2003-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2004-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2004026307-A1
titleOfInvention Triazole derivatives as transforming growth factor (tgf) inhibitors
abstract Novel triazole derivatives of formula (Ia-c) intermediates for their preparation, pharmaceutical compositions containing them and their medicinal use are described. The compounds of the present invention are potent inhibitors of transforming growth factor ('TGF')-βsignaling pathway. They are useful in the treatment of various TGF-related disease states including, for example, cancer and fibrotic diseases.
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Total number of triples: 569.