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filingDate 2003-07-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_823fb9a986db1372fdcff7f7543c5d31
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f06d39f13c9b110b0cf11195fc6f8ad9
publicationDate 2004-01-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2004009625-A2
titleOfInvention PEPTIDES AND PEPTIDE DERIVATIVES FOR THE TREATMENT OF α-SYNUCLEIN-RELATED DISEASES
abstract The invention provides peptides which comprise a sequence of three to twelve contiguous amino acid residues (the 'contiguous sequence') from amino acid residues 61 to 100 of naturally occurring α-synuclein. The contiguous sequence is linked at its N-terminal and/or C-terminal end to one or more further amino acid residue(s) which are more hydrophilic than the amino acid residue to which that end of the sequence is linked in naturally occurring α-synuclein. The invention also provides derivatives and analogues of such peptides. Peptides, derivatives or analogues of the invention are of use in prevention of α-synuclein oligomerisation and/or aggregation associated with the diseases known as the synucleinopathies. As a result peptides according to the invention are susceptible of use in the preparation of medicaments, and also in methods of treatment, for prevention and/or treatment of synucleinopathies.
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