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filingDate 2003-03-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-10-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03084954-A1
titleOfInvention Tropane derivatives as ccr5 modulators
abstract The present invention provides compounds of formula (I) wherein, X, Y, R1, R2 and R2 are as defined hereinabove. The compounds of the present invention are modulators, especially antagonists, of the activity of chemokine CCR5 receptors. Modulators of the CCR5 receptor may be useful in the treatment of various inflammatory diseases and conditions, and in the treatment of infection by HIV and genetically related retroviruses.
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Total number of triples: 822.