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filingDate 2003-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2005-02-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0bd2edb68c61c37cbb2f31237fe7d1e0
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ec512dffe1118260972d1991ac7f377a
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publicationDate 2005-02-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6855724-B2
titleOfInvention Tropane derivatives useful in therapy
abstract The present invention provides compounds of formula (I) n n nwherein X, Y, R 1 , R 2 and R 3 are as defined hereinabove.n n The compounds of the present invention are modulators, especially antagonists, of the activity of chemokine CCR5 receptors. Modulators of the CCR5 receptor may be useful in the treatment of various inflammatory diseases and conditions, and in the treatment of infection by HIV and genetically related retroviruses.
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Total number of triples: 1209.