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filingDate 2001-03-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7b2b217842f102e2ab22651fa1abac2c
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publicationDate 2001-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0164939-A2
titleOfInvention Process for obtaining inhibitors/activators of an enzyme
abstract The invention relates of a generally applicable process for obtaining inhibitors/activators of an enzyme by using a mutant enzyme that binds but is enzymatically inactive using a fluorescence polarization based or other method to measure protein-protein interaction. The obtained inhibitors/activators can be used for the preparation of medicaments for treating diseases caused by or involved with the activity of the enzyme.
priorityDate 2000-03-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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