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filingDate 2016-11-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2f14706fa730a7d207793842f3906bdf
publicationDate 2018-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9975891-B2
titleOfInvention Lactam-containing compounds and derivatives thereof as factor Xa inhibitors
abstract The present application describes lactam-containing compounds and derivatives thereof of Formula I:n nP 4 —P-M-M 4   In nor pharmaceutically acceptable salt forms thereof, wherein ring P, if present is a 5-7 membered carbocycle or heterocycle and ring M is a 5-7 membered carbocycle or heterocycle. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.
priorityDate 2001-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 3969.